BU08028 [Ligand Id: 9294] activity data from GtoPdb

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  • δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
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  • κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
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  • μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
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  • NOP receptor in Human [GtoPdb: 320] [UniProtKB: P41146]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
GtoPdb - - 8.8 pKi 1.59 nM Ki J Pharmacol Exp Ther (2011) 336: 952-61 [PMID:21177476]
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
GtoPdb - - 8.25 pKi 5.63 nM Ki J Pharmacol Exp Ther (2011) 336: 952-61 [PMID:21177476]
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
GtoPdb - - 8.67 pKi 2.14 nM Ki J Pharmacol Exp Ther (2011) 336: 952-61 [PMID:21177476]
NOP receptor in Human [GtoPdb: 320] [UniProtKB: P41146]
GtoPdb - - 8.07 pKi 8.46 nM Ki J Pharmacol Exp Ther (2011) 336: 952-61 [PMID:21177476]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.