VER-246608 [Ligand Id: 9350] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| pyruvate dehydrogenase kinase 2 in Human [GtoPdb: 2142] [UniProtKB: Q15119] | ||||||||
| GtoPdb | In vitro functional assay | - | 7.08 | pIC50 | 84 | nM | IC50 | Oncotarget (2014) 5: 12862-76 [PMID:25404640] |
| pyruvate dehydrogenase kinase 3 in Human [GtoPdb: 2143] [UniProtKB: Q15120] | ||||||||
| GtoPdb | In vitro functional assay | - | 7.4 | pIC50 | 40 | nM | IC50 | Oncotarget (2014) 5: 12862-76 [PMID:25404640] |
| pyruvate dehydrogenase kinase 4 in Human [GtoPdb: 2144] [UniProtKB: Q16654] | ||||||||
| GtoPdb | In vitro functional assay | - | 7.04 | pIC50 | 91 | nM | IC50 | Oncotarget (2014) 5: 12862-76 [PMID:25404640] |
| pyruvate dehydrogenase kinase 1 in Human [GtoPdb: 2915] [UniProtKB: Q15118] | ||||||||
| GtoPdb | In vitro functional assay | - | 7.46 | pIC50 | 35 | nM | IC50 | Oncotarget (2014) 5: 12862-76 [PMID:25404640] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
