GSK143 [Ligand Id: 9388] activity data from GtoPdb

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  • aurora kinase A in Human [GtoPdb: 1936] [UniProtKB: O14965]
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  • spleen associated tyrosine kinase in Human [GtoPdb: 2230] [UniProtKB: P43405]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
aurora kinase A in Human [GtoPdb: 1936] [UniProtKB: O14965]
GtoPdb Enzyme inhibition assay using recombinant human protein - 8.32 pIC50 4.8 nM IC50 Bioorg Med Chem Lett (2011) 21: 6188-94 [PMID:21903390]
spleen associated tyrosine kinase in Human [GtoPdb: 2230] [UniProtKB: P43405]
GtoPdb Enzyme inhibition assay using recombinant human protein - 8.12 pIC50 7.5 nM IC50 Bioorg Med Chem Lett (2011) 21: 6188-94 [PMID:21903390]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.