fruquintinib [Ligand Id: 9428] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fms related receptor tyrosine kinase 1 in Human [GtoPdb: 1812] [UniProtKB: P17948] | ||||||||
| GtoPdb | Evaluated in a [32]p-ATP incorporation assay | - | 7.48 | pIC50 | 33 | nM | IC50 | Cancer Biol Ther (2014) 15: 1635-45 [PMID:25482937] |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | Evaluated in a [32]p-ATP incorporation assay | - | 7.46 | pIC50 | 35 | nM | IC50 | Cancer Biol Ther (2014) 15: 1635-45 [PMID:25482937] |
| GtoPdb | Evaluated in a Z-lyte assay. | - | 7.6 | pIC50 | 25 | nM | IC50 | Cancer Biol Ther (2014) 15: 1635-45 [PMID:25482937] |
| fms related receptor tyrosine kinase 4 in Human [GtoPdb: 1814] [UniProtKB: P35916] | ||||||||
| GtoPdb | Evaluated in a [32]p-ATP incorporation assay | - | 9.3 | pIC50 | 0.5 | nM | IC50 | Cancer Biol Ther (2014) 15: 1635-45 [PMID:25482937] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
