Lys[Z(NO2)]-Val [Ligand Id: 9486] activity data from GtoPdb

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  • Peptide transporter 1 in Human [GtoPdb: 984] [UniProtKB: P46059]
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  • Peptide transporter 2 in Human [GtoPdb: 985] [UniProtKB: Q16348]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Peptide transporter 1 in Human [GtoPdb: 984] [UniProtKB: P46059]
GtoPdb Competition assays in Caco-2 cells expressing PEPT1. - 5.7 pKi 2000 nM Ki Eur J Pharm Sci (2004) 21: 61-7 [PMID:14706812]
Peptide transporter 2 in Human [GtoPdb: 985] [UniProtKB: Q16348]
GtoPdb - - 7 pKi - - - Amino Acids (2006) 31: 137-56 [PMID:16868651];
J Biol Chem (2002) 277: 7287-92 [PMID:11751927]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.