glycyl-sarcosine [Ligand Id: 9505] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL175737 (Glycylsarcosine, Gly-Sar, Gly-Sarcosin)
  • Peptide transporter 2/Solute carrier family 15 member 2 in Human [ChEMBL: CHEMBL1743125] [GtoPdb: 985] [UniProtKB: Q16348]
  • This target only has 1 pki data point
  • 4.19
1 CHEMBL175737_lig_chart_1 Solute carrier family 15 member 2 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Peptide transporter 2/Solute carrier family 15 member 2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1743125] [GtoPdb: 985] [UniProtKB: Q16348]
ChEMBL TP_TRANSPORTER: inhibition of Cephalexin uptake in SKPT cells F 4.19 pKi 64000 nM Ki J. Biol. Chem. (1995) 270: 25672-25677 [PMID:7592745]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]