GSK8814 [Ligand Id: 9521] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ATPase family AAA domain containing 2 in Human [GtoPdb: 2719] [UniProtKB: Q6PL18] | ||||||||
| GtoPdb | By isothermal titration calorimetry (ICT) assay. | - | 8.1 | pKd | 8 | nM | Kd | Angew Chem Int Ed Engl (2016) 55: 11382-6 [PMID:27530368] |
| GtoPdb | By Bromosphere assay using full length endogenous protein. | - | 8.9 | pKi | 1.25 | nM | Ki | Angew Chem Int Ed Engl (2016) 55: 11382-6 [PMID:27530368] |
| GtoPdb | By TR-FRET assay. | - | 7.3 | pIC50 | 50.1 | nM | IC50 | Angew Chem Int Ed Engl (2016) 55: 11382-6 [PMID:27530368] |
| ATPase family AAA domain containing 2B in Human [GtoPdb: 2720] [UniProtKB: Q9ULI0] | ||||||||
| GtoPdb | By TR-FRET assay. | - | 7.7 | pIC50 | 19.9 | nM | IC50 | Angew Chem Int Ed Engl (2016) 55: 11382-6 [PMID:27530368] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
