eganelisib [Ligand Id: 9563] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | - | - | 7.77 | pKd | 17 | nM | Kd | ACS Med Chem Lett (2016) 7: 862-7 [PMID:27660692] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | - | - | 7.09 | pKd | 82 | nM | Kd | ACS Med Chem Lett (2016) 7: 862-7 [PMID:27660692] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | - | - | 7.64 | pKd | 23 | nM | Kd | ACS Med Chem Lett (2016) 7: 862-7 [PMID:27660692] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | - | - | 9.54 | pKd | 0.29 | nM | Kd | ACS Med Chem Lett (2016) 7: 862-7 [PMID:27660692] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
