SR8185 [Ligand Id: 9578] activity data from GtoPdb

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  • inhibitor of nuclear factor kappa B kinase subunit epsilon in Human [GtoPdb: 2040] [UniProtKB: Q14164]
  • This target only has 0 pki data point
1 _lig_chart_1 inhibitor of nuclear factor kappa B kinase subunit epsilon Human
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  • TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2]
  • This target only has 0 pki data point
2 _lig_chart_2 TANK binding kinase 1 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
inhibitor of nuclear factor kappa B kinase subunit epsilon in Human [GtoPdb: 2040] [UniProtKB: Q14164]
GtoPdb In an enzyme assay. - 8.52 pIC50 3 nM IC50 Int. J. Cancer (2014) 134: 1972-80 [PMID:24150799]
TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2]
GtoPdb In an enzyme assay. - 8 pIC50 <10 nM IC50 Int. J. Cancer (2014) 134: 1972-80 [PMID:24150799]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.