andrographolide [Ligand Id: 9675] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • TAS2R8 in Human [GtoPdb: 664] [UniProtKB: Q9NYW2]
There should be some charts here, you may need to enable JavaScript!
  • TAS2R50 in Human [GtoPdb: 677] [UniProtKB: P59544]
There should be some charts here, you may need to enable JavaScript!
  • TAS2R46 in Human [GtoPdb: 679] [UniProtKB: P59540]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TAS2R8 in Human [GtoPdb: 664] [UniProtKB: Q9NYW2]
GtoPdb - - 3.96 pEC50 110000 nM EC50 J Med Chem (2020) 63: 4957-4977 [PMID:32330040]
TAS2R50 in Human [GtoPdb: 677] [UniProtKB: P59544]
GtoPdb - - 4.64 pEC50 22900 nM EC50 J Agric Food Chem (2009) 57: 9860-6 [PMID:19817411]
TAS2R46 in Human [GtoPdb: 679] [UniProtKB: P59540]
GtoPdb - - 4.89 pEC50 13000 nM EC50 PLoS Genet (2015) 11: e1005530 [PMID:26406243]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.