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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345] | ||||||||
GtoPdb | In an in vitro enzymatic assay. | - | 5.25 | pIC50 | 5560 | nM | IC50 | ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499] |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
GtoPdb | In an in vitro enzymatic assay. | - | 6.07 | pIC50 | 856 | nM | IC50 | ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499] |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
GtoPdb | In an in vitro enzymatic assay. | - | 6.06 | pIC50 | 867 | nM | IC50 | ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499] |
serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716] | ||||||||
GtoPdb | In an in vitro enzymatic inhibition assay. | - | 6.53 | pIC50 | 295 | nM | IC50 | ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.