tropifexor [Ligand Id: 9725] activity data from GtoPdb

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  • Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
GtoPdb In a HTRF assay. - 9.7 pEC50 0.2 nM EC50 J Med Chem (2017) 60: 9960-9973 [PMID:29148806]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.