BMS-986187 [Ligand Id: 9748] activity data from GtoPdb

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  • δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
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  • μ receptor in Rat [GtoPdb: 319] [UniProtKB: P33535]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
GtoPdb - - 8.15 pKi 7 nM Ki
μ receptor in Rat [GtoPdb: 319] [UniProtKB: P33535]
GtoPdb - - 7.2 pKi 63 nM Ki Mol Pharmacol (2018) 93: 157-167 [PMID:29233847]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.