SAR-20347 [Ligand Id: 9803] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | In a TR-FRET assay. | - | 7.23 | pIC50 | 59 | nM | IC50 | J Immunol (2014) 193: 3278-87 [PMID:25156366] |
| GtoPdb | In a 33P-ATP assay. | - | 7.64 | pIC50 | 23 | nM | IC50 | J Immunol (2014) 193: 3278-87 [PMID:25156366] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | In a TR-FRET assay. | - | 6.05 | pIC50 | 882 | nM | IC50 | J Immunol (2014) 193: 3278-87 [PMID:25156366] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | In a TR-FRET assay. | - | 5.84 | pIC50 | 1437 | nM | IC50 | J Immunol (2014) 193: 3278-87 [PMID:25156366] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | In a TR-FRET assay. | - | 7.89 | pIC50 | 13 | nM | IC50 | J Immunol (2014) 193: 3278-87 [PMID:25156366] |
| GtoPdb | In a 33P-ATP assay. | - | 9.22 | pIC50 | 0.6 | nM | IC50 | J Immunol (2014) 193: 3278-87 [PMID:25156366] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
