LIMKi3 [Ligand Id: 9839] activity data from GtoPdb

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  • LIM domain kinase 1 in Human [GtoPdb: 2054] [UniProtKB: P53667]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 LIM domain kinase 1 Human
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  • LIM domain kinase 2 in Human [GtoPdb: 2055] [UniProtKB: P53671]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 LIM domain kinase 2 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
LIM domain kinase 1 in Human [GtoPdb: 2054] [UniProtKB: P53667]
GtoPdb - - 8.15 pIC50 7 nM IC50 Br J Pharmacol (2018) 175: 2077-2096 [PMID:29574791];
Mol Cancer Ther (2008) 7: 3490-8 [PMID:19001433];
J Cell Biol (2010) 191: 169-85 [PMID:20876278];
J Neurosci (2012) 32: 5284-97 [PMID:22496574]
LIM domain kinase 2 in Human [GtoPdb: 2055] [UniProtKB: P53671]
GtoPdb - - 8.1 pIC50 8 nM IC50 Br J Pharmacol (2018) 175: 2077-2096 [PMID:29574791];
Mol Cancer Ther (2008) 7: 3490-8 [PMID:19001433];
J Cell Biol (2010) 191: 169-85 [PMID:20876278];
J Neurosci (2012) 32: 5284-97 [PMID:22496574]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.