apilimod [Ligand Id: 9859] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphoinositide kinase, FYVE-type zinc finger containing in Human [GtoPdb: 2857] [UniProtKB: Q9Y2I7] | ||||||||
| GtoPdb | Binding constant for Cy5-apilimod to PIKfyve kinase domain. | - | 7.19 | pKd | 65 | nM | Kd | Chem Biol (2013) 20: 912-21 [PMID:23890009] |
| GtoPdb | Effect of apilimod on hPIKfyve kinase activity in vitro measuringPI(3)P conversion to PI(3,5)P2. | - | 7.85 | pIC50 | 14 | nM | IC50 | Chem Biol (2013) 20: 912-21 [PMID:23890009] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
