Synonyms: L-084 | LJC 11,084 | LJC-11,084 | LJC-11084 | Orapenem® | TBPM-PI
tebipenem pivoxil is an approved drug (Japan)
Compound class:
Synthetic organic
Comment: Tebipenem pivoxil is an orally available pivaloyloxymethyl ester prodrug of the β-lactam antibacterial tebipenem [1-2]. The ester bond is cleaved, releasing active tebipenem (PubChem CID 9800194; LJC-11036). The drug has Gram-negative activity. Tebipenem pivoxil hydrobromide (SPR994) is another formulation of the same drug.
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Classification | |
Compound class | Synthetic organic |
Approved drug? | Yes (Japan) |
IUPAC Name |
2,2-dimethylpropanoyloxymethyl (4R,5S,6S)-3-[1-(4,5-dihydro-1,3-thiazol-2-yl)azetidin-3-yl]sulfanyl-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylate |
International Nonproprietary Names | |
INN number | INN |
7924 | tebipenem pivoxil |
Synonyms |
L-084 | LJC 11,084 | LJC-11,084 | LJC-11084 | Orapenem® | TBPM-PI |
Database Links | |
Specialist databases | |
Antibiotic DB | Tebipenem |
Other databases | |
CAS Registry No. | 161715-24-8 (source: WHO INN record) |
DrugCentral Ligand | 2574 |
GtoPdb PubChem SID | 405560305 |
PubChem CID | 9892071 |
Search Google for chemical match using the InChIKey | SNUDIPVBUUXCDG-QHSBEEBCSA-N |
Search Google for chemicals with the same backbone | SNUDIPVBUUXCDG |
Search PubMed clinical trials | tebipenem pivoxil |
Search PubMed titles | tebipenem pivoxil |
Search PubMed titles/abstracts | tebipenem pivoxil |
UniChem Compound Search for chemical match using the InChIKey | SNUDIPVBUUXCDG-QHSBEEBCSA-N |
UniChem Connectivity Search for chemical match using the InChIKey | SNUDIPVBUUXCDG-QHSBEEBCSA-N |