Synonyms: [3H]-U69593
Compound class:
Synthetic organic
Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
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References |
1. Lahti RA, Mickelson MM, McCall JM, Von Voigtlander PF. (1985)
[3H]U-69593 a highly selective ligand for the opioid kappa receptor. Eur J Pharmacol, 109 (2): 281-4. [PMID:2986999] |
2. Payza K. (2003)
Binding and activity of opioid ligands at the cloned human delta, mu and kappa receptors. In The Delta Receptor Edited by Chang KJ (CRC Press) 261-275. [ISBN:0824740319] |
3. Simonin F, Gavériaux-Ruff C, Befort K, Matthes H, Lannes B, Micheletti G, Mattéi MG, Charron G, Bloch B, Kieffer B. (1995)
kappa-Opioid receptor in humans: cDNA and genomic cloning, chromosomal assignment, functional expression, pharmacology, and expression pattern in the central nervous system. Proc Natl Acad Sci USA, 92 (15): 7006-10. [PMID:7624359] |