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BIM 23023   Click here for help

GtoPdb Ligand ID: 2032

Compound class: Peptide
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Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 9.4 pKi - 2
pKi 9.4 [2]
SST2 receptor Rn Agonist Full agonist 9.2 pKi - 1
pKi 9.2 [1]
SST5 receptor Hs Agonist Full agonist 8.4 – 9.4 pKi - 1-2
pKi 8.4 – 9.4 [1-2]
SST2 receptor Mm Agonist Full agonist 7.0 – 9.4 pKi - 1
pKi 7.0 – 9.4 [1]
SST3 receptor Hs Agonist Full agonist 8.1 pKi - 2
pKi 8.1 [2]
SST5 receptor Rn Agonist Full agonist 7.8 pKi - 1
pKi 7.8 [1]
SST3 receptor Rn Agonist Full agonist 7.0 pKi - 1
pKi 7.0 [1]
SST3 receptor Mm Agonist Full agonist 7.9 pIC50 - 3
pIC50 7.9 [3]