Kir5.1
|
|
|
Rn |
Channel blocker |
Antagonist |
- |
- |
3x10-3 |
28 |
|
⤷ |
Conc range: 3x10-3 M
Kir5.1 expressed with PSD-95
[28]
Voltage:
-120.0 – 20.0 mV
|
K2P18.1
|
|
|
N/A |
Channel blocker |
- |
- |
- |
2.5x10-3 - 3x10-3 |
|
|
⤷ |
Conc range: 2.5x10-3 - 3x10-3 M
|
K2P4.1
|
|
|
Rn |
Channel blocker |
- |
- |
- |
2x10-3 |
10 |
|
⤷ |
Conc range: 2x10-3 M
[10]
|
Kir1.1
|
|
|
Hs |
Channel blocker |
Antagonist |
- |
- |
1x10-3 |
24 |
|
⤷ |
Conc range: 1x10-3 M
[24]
Voltage:
-160.0 – 80.0 mV
|
K2P16.1
|
|
|
Hs |
Channel blocker |
- |
- |
- |
1x10-3 |
5 |
|
⤷ |
Conc range: 1x10-3 M
[5]
|
Kir4.1
|
|
|
Rn |
Channel blocker |
Antagonist |
- |
- |
3x10-6 - 1x10-3 |
11,27,29 |
|
⤷ |
Conc range: 3x10-6 - 1x10-3 M
[11,27,29]
Voltage:
-160.0 – 60.0 mV
|
Kir3.1
|
|
|
Hs |
Channel blocker |
Antagonist |
- |
- |
1x10-4 - 3x10-4 |
23 |
|
⤷ |
Conc range: 1x10-4 - 3x10-4 M
[23]
Voltage:
Physiological
|
Kir3.1
|
|
|
Rn |
Channel blocker |
Antagonist |
- |
- |
1x10-4 - 2.5x10-4 |
3 |
|
⤷ |
Conc range: 1x10-4 - 2.5x10-4 M
[3]
Voltage:
Physiological
|
Kir4.2
|
|
|
Mm |
Channel blocker |
Antagonist |
- |
- |
1x10-5 - 1x10-4 |
21 |
|
⤷ |
Conc range: 1x10-5 - 1x10-4 M
Kir4.2 expressed in Xenopus oocytes
[21]
Voltage:
-120.0 – 100.0 mV
|
Kir2.2
|
|
|
Mm |
Gating inhibitor |
Antagonist |
- |
- |
5x10-5 |
26 |
|
⤷ |
Conc range: 5x10-5 M
[26]
Voltage:
-150.0 – -50.0 mV
|
Kir2.1
|
|
|
Mm |
Channel blocker |
Antagonist |
3.9 – 5.6 |
pKd |
1x10-6 - 1x10-4 |
1 |
|
⤷ |
pKd
3.9 – 5.6
Conc range: 1x10-6 - 1x10-4 M
[1]
Voltage:
0.0 – -80.0 mV
|
Kir2.4
|
|
|
Hs |
Channel blocker |
Antagonist |
3.3 |
pKd |
- |
9 |
|
⤷ |
pKd
3.3
[9]
Voltage:
0.0 mV
|
Kv2.1
|
|
|
Rn |
Channel blocker (Extracellular Ba2+) |
- |
1.5 – 4.9 |
pKd |
- |
25 |
|
⤷ |
pKd
4.9
[25]
pKd
1.5
[25]
|
Kir2.2
|
|
|
Rn |
Gating inhibitor |
Antagonist |
5.2 |
pKi |
- |
32 |
|
⤷ |
pKi
5.2
[32]
Voltage:
-80.0 mV
|
Kir2.4
|
|
|
Rn |
Channel blocker |
Antagonist |
3.4 – 4.2 |
pKi |
1x10-6 - 1x10-3 |
31-32 |
|
⤷ |
pKi
3.4 – 4.2
Conc range: 1x10-6 - 1x10-3 M
[31-32]
Voltage:
-80.0 – -100.0 mV
|
Kir7.1
|
|
|
Hs |
Channel blocker |
Antagonist |
3.2 |
pKi |
- |
4,13-14,19 |
|
⤷ |
pKi
3.2
[4,13-14,19]
Voltage:
-100.0 mV
|
Kir3.4
|
|
|
Rn |
Channel blocker |
Antagonist |
3.3 |
pEC50 |
- |
12 |
|
⤷ |
pEC50
3.3
[12]
Voltage:
-80.0 mV
|
Kir2.3
|
|
|
Mm |
Channel blocker |
Antagonist |
5.2 |
pIC50 |
5x10-6 - 5x10-4 |
16,18 |
|
⤷ |
pIC50
5.2
Conc range: 5x10-6 - 5x10-4 M
[16,18]
Voltage:
-150.0 mV
|
Kir2.3
|
|
|
Hs |
Channel blocker |
Antagonist |
5.0 |
pIC50 |
3x10-6 - 5x10-4 |
17,22,30 |
|
⤷ |
pIC50
5.0
Conc range: 3x10-6 - 5x10-4 M
[17,22,30]
Voltage:
-60.0 mV
|
Kir3.1
|
|
|
Rn |
Channel blocker |
Antagonist |
4.7 |
pIC50 |
- |
3 |
|
⤷ |
pIC50
4.7
Kir3.1 expressed in Xenopus oocytes
[3]
|
Kv12.1
|
|
|
Hs |
Channel blocker |
- |
3.7 |
pIC50 |
- |
34 |
|
⤷ |
pIC50
3.7
[34]
|
Kir1.1
|
|
|
Rn |
Channel blocker |
Antagonist |
2.3 – 4.2 |
pIC50 |
1x10-4 |
8,33 |
|
⤷ |
pIC50
2.3 – 4.2
Conc range: 1x10-4 M
[8,33]
Voltage:
0.0 – -100.0 mV
|
KNa1.2
|
|
|
Hs |
Channel blocker |
Inhibition |
3.0 |
pIC50 |
- |
2 |
|
⤷ |
pIC50
3.0
[2]
|
Kv1.8
|
|
|
Hs |
Channel blocker |
- |
2.3 |
pIC50 |
- |
15 |
|
⤷ |
pIC50
2.3
[15]
|
K2P3.1
|
|
|
Hs |
Channel blocker |
- |
0.3 |
pIC50 |
- |
|
|
⤷ |
pIC50
0.3
|
K2P6.1
|
|
|
Rn |
Channel blocker |
- |
- |
pIC50 |
1x10-5 - 1x10-4 |
20 |
|
⤷ |
pIC50
Conc range: 1x10-5 - 1x10-4 M
[20]
|
K2P13.1
|
|
|
N/A |
Channel blocker |
- |
- |
- |
- |
|
|
⤷ |
|