Synonyms: compound 2 [PMID: 18281931] | EVG | GS-9137 | GS9137 | JTK-303 | JTK303 | Vitekta®
elvitegravir is an approved drug (EMA (2013), FDA (2014), UK (2021))
Compound class:
Synthetic organic
Comment: Elvitegravir (GS-9137) is an HIV integrase inhibitor antiretroviral drug [1].
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Bioactivity Comments |
Elvitegravir (GS-9137) inhibits HIV integrase-mediated strand transfer with an IC50 of 7.2 nM [1]. Its antiviral EC50 is is 0.9 nM. |