[125I]Hpp-desArg10HOE140   Click here for help

GtoPdb Ligand ID: 3791

Synonyms: [125I]-Hpp-desArg9HOE140
 Ligand is labelled  Ligand is radioactive
Comment: Radiolabelled analogue of icatibant (HOE 140), a synthetic analogue of bradykinin.
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Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
B1 receptor Hs Antagonist Antagonist 10.0 pKd - 1-2
pKd 10.0 (Kd 1x10-10 M)
pKd 10.0 (Kd 1x10-10 M) [1-2]