[D-Tyr6,Apa-4Cl11,Phe13,Nle14]bombesin-(6-14)   Click here for help

GtoPdb Ligand ID: 3946

Synonyms: [D-Tyr6,Apa-4Cl11,Phe13,Nle14]bombesin6-14
Comment: Synthetic analogue of bombesin
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
BB3 receptor Hs Agonist Full agonist 8.1 pKi - 2
pKi 8.1 (Ki 8x10-9 M) [2]
BB3 receptor Hs Agonist Full agonist 7.4 – 8.9 pIC50 - 1,3
pIC50 7.4 – 8.9 (IC50 4x10-8 – 1.4x10-9 M) [1,3]