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[D-Tyr6,Apa-4Cl11,Phe13,Nle14]bombesin-(6-14)   Click here for help

GtoPdb Ligand ID: 3946

Synonyms: [D-Tyr6,Apa-4Cl11,Phe13,Nle14]bombesin6-14
Compound class: Peptide
Comment: Synthetic analogue of bombesin
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Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
BB3 receptor Hs Agonist Full agonist 8.1 pKi - 2
pKi 8.1 (Ki 8x10-9 M) [2]
BB3 receptor Hs Agonist Full agonist 7.4 – 8.9 pIC50 - 1,3
pIC50 7.4 – 8.9 (IC50 4x10-8 – 1.4x10-9 M) [1,3]