[125I][Tyr26]galanin (pig)

Ligand id: 6117

Name: [125I][Tyr26]galanin (pig)    

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
GAL1 receptor Rn Agonist Agonist 9.5 – 10.7 pKd - 2-4,6-8
pKd 9.5 – 10.7 (Kd 3x10-10 – 1.9x10-11 M) Two populations of binding sites have been identified in transfected cells with Kds of 0.3 and 0.019nM. [2-4,6-8]
GAL1 receptor Hs Agonist Agonist 9.8 pKd - 1
pKd 9.8 (Kd 1.5x10-10 M) [1]
GAL2 receptor Hs Agonist Agonist 9.5 – 9.9 pKd - 1,4
pKd 9.9 (Kd 1.2x10-10 M) [4]
pKd 9.5 (Kd 3.1x10-10 M) [1]
GAL2 receptor Rn Agonist Agonist 8.4 – 9.9 pKd - 3,5,8-9
pKd 8.4 – 9.9 (Kd 4x10-9 – 1.3x10-10 M) [3,5,8-9]
GAL3 receptor Rn Agonist Agonist 9.0 – 9.3 pKd - 8,10
pKd 9.0 – 9.3 (Kd 9.7x10-10 – 5.5x10-10 M) [8,10]
GAL3 receptor Hs Agonist Agonist 8.6 pKd - 1,8
pKd 8.6 (Kd 2.24x10-9 M) [1,8]