poziotinib

poziotinib selectivity at human targets
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Target Value Parameter Concentration range (M) Type Action
erb-b2 receptor tyrosine kinase 2 8.3 pIC50 - Inhibitor Inhibition
epidermal growth factor receptor 8.1 pIC50 - Inhibitor Inhibition
erb-b2 receptor tyrosine kinase 4 7.6 pIC50 - Inhibitor Inhibition