INN: valsartan Comments: Valsartan is an antagonist with high affinity for the type I (AT1) angiotensin receptor. Clinical use: valsartan (80mg) was approved by the FDA in June 2016 for the treatment of hypertension
Antagonists - comment: valsartan, EXP3174, azilsartan medoxomil and saprisartan are all classed as insurmountable antagonists.Partial agonist: Activate the receptor