nidufexor [Ligand Id: 10655] activity data from GtoPdb

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  • Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
GtoPdb Determined in a HTRF FXR coactivator interaction assay using GST-tagged hFXR ligand binding domain and biotinylated SRC-1 peptide. - 9.3 pEC50 0.5 nM EC50 J Med Chem (2020) 63: 3868-3880 [PMID:31940200]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.