TP0556351 [Ligand Id: 12057] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| MMP2 in Human [GtoPdb: 1629] [UniProtKB: P08253] | ||||||||
| GtoPdb | - | - | 9.7 | pIC50 | 0.2 | nM | IC50 | J Med Chem (2022) 65: 8493-8510 [PMID:35687819] |
| MMP8 in Human [GtoPdb: 1632] [UniProtKB: P22894] | ||||||||
| GtoPdb | - | - | 5.43 | pIC50 | 3725 | nM | IC50 | J Med Chem (2022) 65: 8493-8510 [PMID:35687819] |
| MMP9 in Human [GtoPdb: 1633] [UniProtKB: P14780] | ||||||||
| GtoPdb | - | - | 5.07 | pIC50 | 8508 | nM | IC50 | J Med Chem (2022) 65: 8493-8510 [PMID:35687819] |
| MMP12 in Human [GtoPdb: 1636] [UniProtKB: P39900] | ||||||||
| GtoPdb | - | - | 5.86 | pIC50 | 1367 | nM | IC50 | J Med Chem (2022) 65: 8493-8510 [PMID:35687819] |
| MMP13 in Human [GtoPdb: 1637] [UniProtKB: P45452] | ||||||||
| GtoPdb | - | - | 6.76 | pIC50 | 174 | nM | IC50 | J Med Chem (2022) 65: 8493-8510 [PMID:35687819] |
| MMP14 in Human [GtoPdb: 1638] [UniProtKB: P50281] | ||||||||
| GtoPdb | - | - | 5.65 | pIC50 | 2216 | nM | IC50 | J Med Chem (2022) 65: 8493-8510 [PMID:35687819] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
