NNMT inhibitor 14 [PMID: 35904556] [Ligand Id: 12166] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| nicotinamide N-methyltransferase in Human [GtoPdb: 3205] [UniProtKB: P40261] | ||||||||
| GtoPdb | Determined in a cell-based assay, with hNNMT expressed in HEK293 cells | - | 6.4 | pIC50 | 400 | nM | IC50 | J Med Chem (2022) 65: 10655-10673 [PMID:35904556] |
| GtoPdb | Determined in a cell-free assay system | - | 8.96 | pIC50 | 1.1 | nM | IC50 | J Med Chem (2022) 65: 10655-10673 [PMID:35904556] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
