LY3540378 [Ligand Id: 12502] activity data from GtoPdb

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  • RXFP1 in Monkey [GtoPdb: 351]
  • RXFP1 in Human [GtoPdb: 351] [UniProtKB: Q9HBX9]
  • RXFP1 in Mouse [GtoPdb: 351] [UniProtKB: Q6R6I7]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
RXFP1 in Monkey [GtoPdb: 351]
GtoPdb Binding affinity determined by SPR. - 10.4 pKd 0.04 nM Kd Br J Pharmacol (2023) 180: 1965-1980 [PMID:36780899]
RXFP1 in Human [GtoPdb: 351] [UniProtKB: Q9HBX9]
GtoPdb Binding affinity determined by SPR. - 10.09 pKd 0.08 nM Kd Br J Pharmacol (2023) 180: 1965-1980 [PMID:36780899]
RXFP1 in Mouse [GtoPdb: 351] [UniProtKB: Q6R6I7]
GtoPdb Binding affinity determined by SPR. - 8.7 pKd 2 nM Kd Br J Pharmacol (2023) 180: 1965-1980 [PMID:36780899]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.