PTD10 [Ligand Id: 12687] activity data from GtoPdb

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  • Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
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  • cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
GtoPdb Inhibition of BTK catalytic activity in a cellular assay - 7.01 pIC50 97 nM IC50 Journal of Mediconal Chemistry (2023) :
cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2]
GtoPdb Measuring target engagement in a NanoBRET competitive displacement assay. - 6.97 pIC50 107 nM IC50 Journal of Mediconal Chemistry (2023) :

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.