tegeprotafib [Ligand Id: 12884] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| protein tyrosine phosphatase non-receptor type 1 in Human [GtoPdb: 2976] [UniProtKB: P18031] | ||||||||
| GtoPdb | Determined in a mobility shift assays using a phosphorylated insulin receptor peptide as substrate to measure inhibition of PTPN1-mediated dephopshorylation | - | 9 | pIC50 | 1 | nM | IC50 | WO2021127499A1. Protein tyrosine phosphatase inhibitors and methods of use thereof (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
