HPG1860 [Ligand Id: 12910] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
GtoPdb Determined in a TR-FRET based FXR bioactivity assay - 8.3 pEC50 5 nM EC50 J Med Chem (2023) 66: 9363-9375 [PMID:37424079]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.