PF-9363 [Ligand Id: 12938] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • lysine acetyltransferase 5 in Human [GtoPdb: 2664] [UniProtKB: Q92993]
There should be some charts here, you may need to enable JavaScript!
  • lysine acetyltransferase 6A in Human [GtoPdb: 2665] [UniProtKB: Q92794]
There should be some charts here, you may need to enable JavaScript!
  • lysine acetyltransferase 6B in Human [GtoPdb: 2666] [UniProtKB: Q8WYB5]
There should be some charts here, you may need to enable JavaScript!
  • lysine acetyltransferase 7 in Human [GtoPdb: 2667] [UniProtKB: O95251]
There should be some charts here, you may need to enable JavaScript!
  • lysine acetyltransferase 8 in Human [GtoPdb: 2668] [UniProtKB: Q9H7Z6]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
lysine acetyltransferase 5 in Human [GtoPdb: 2664] [UniProtKB: Q92993]
GtoPdb - - 6.38 pIC50 420 nM IC50 Cell Chem Biol (2023) 30: 1191-1210.e20 [PMID:37557181]
lysine acetyltransferase 6A in Human [GtoPdb: 2665] [UniProtKB: Q92794]
GtoPdb - - 9.57 pIC50 0.27 nM IC50 Cell Chem Biol (2023) 30: 1191-1210.e20 [PMID:37557181]
lysine acetyltransferase 6B in Human [GtoPdb: 2666] [UniProtKB: Q8WYB5]
GtoPdb - - 8.62 pIC50 2.4 nM IC50 Cell Chem Biol (2023) 30: 1191-1210.e20 [PMID:37557181]
lysine acetyltransferase 7 in Human [GtoPdb: 2667] [UniProtKB: O95251]
GtoPdb - - 7.15 pIC50 70 nM IC50 Cell Chem Biol (2023) 30: 1191-1210.e20 [PMID:37557181]
lysine acetyltransferase 8 in Human [GtoPdb: 2668] [UniProtKB: Q9H7Z6]
GtoPdb - - 6.17 pIC50 670 nM IC50 Cell Chem Biol (2023) 30: 1191-1210.e20 [PMID:37557181]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.