RLY-2608 [Ligand Id: 13065] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | Biochemical inhibition of WT PI3KCA | - | 7.32 | pIC50 | 48 | nM | IC50 | Cancer Discov (2024) 14: 240-257 [PMID:37916956] |
| GtoPdb | Biochemical inhibition of PI3KCA1047R | - | 8.4 | pIC50 | 4 | nM | IC50 | Cancer Discov (2024) 14: 240-257 [PMID:37916956] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
