biKEAP1 [Ligand Id: 13066] activity data from GtoPdb

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  • kelch like ECH-associated protein 1 in Human [GtoPdb: 2757] [UniProtKB: Q14145]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
kelch like ECH-associated protein 1 in Human [GtoPdb: 2757] [UniProtKB: Q14145]
GtoPdb Determined in a fluorescence polarization (FP) assay, measuring displacement of a NRF2 ETGE motif derived peptide from KEAP1 Kelch domain - 8.07 pIC50 8.49 nM IC50 Cell Chem Biol (2023) null: null [PMID:38157852]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.