GNE-235 [Ligand Id: 13104] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| polybromo 1 in Human [GtoPdb: 2738] [UniProtKB: Q86U86] | ||||||||
| GtoPdb | Binding affinity for BD5 of hPBRM1 | - | 4.82 | pKd | 15000 | nM | Kd | J Med Chem (2023) 66: 13116-13134 [PMID:37702400] |
| GtoPdb | Binding affinity for BD2 of hPBRM1 | - | 6.55 | pKd | 280 | nM | Kd | J Med Chem (2023) 66: 13116-13134 [PMID:37702400] |
| SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 2 in Human [GtoPdb: 2739] [UniProtKB: P51531] | ||||||||
| GtoPdb | Binding affinity for hSMARCA2 | - | 5.22 | pKd | 6000 | nM | Kd | J Med Chem (2023) 66: 13116-13134 [PMID:37702400] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
