compound 8a [PMID: 35500474] [Ligand Id: 13121] activity data from GtoPdb

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  • poly(ADP-ribose) polymerase family member 10 in Human [GtoPdb: 3267] [UniProtKB: Q53GL7]
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  • poly(ADP-ribose) polymerase family member 15 in Human [GtoPdb: 3270] [UniProtKB: Q460N3]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
poly(ADP-ribose) polymerase family member 10 in Human [GtoPdb: 3267] [UniProtKB: Q53GL7]
GtoPdb - - 6.85 pIC50 140 nM IC50 Eur J Med Chem (2022) 237: 114362 [PMID:35500474]
poly(ADP-ribose) polymerase family member 15 in Human [GtoPdb: 3270] [UniProtKB: Q460N3]
GtoPdb - - 6.4 pIC50 400 nM IC50 Eur J Med Chem (2022) 237: 114362 [PMID:35500474]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.