CBPD-268 [Ligand Id: 13245] activity data from GtoPdb

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  • CREB binding protein in Human [GtoPdb: 2734] [UniProtKB: Q92793]
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  • E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
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  • cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CREB binding protein in Human [GtoPdb: 2734] [UniProtKB: Q92793]
GtoPdb - - 7.96 pIC50 11 nM IC50 J Med Chem (2024) null: null [PMID:38477974]
E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb - - 8.02 pIC50 9.5 nM IC50 J Med Chem (2024) null: null [PMID:38477974]
cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2]
GtoPdb - - 5.74 pIC50 1800 nM IC50 J Med Chem (2024) null: null [PMID:38477974]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.