CL316243 [Ligand Id: 3462] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1204876 (CL-316243) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| β3-adrenoceptor in Human [GtoPdb: 30] [UniProtKB: P13945] | ||||||||
| GtoPdb | - | - | 5.2 | pKi | - | - | - | Tohoku J Exp Med (2000) 192: 181-93 [PMID:11249148] |
| β3-adrenoceptor in Mouse [GtoPdb: 30] [UniProtKB: P25962] | ||||||||
| GtoPdb | - | - | 5.9 | pKi | - | - | Ki | Mol Pharmacol (2007) 72: 1359-68 [PMID:17717109] |
| GtoPdb | - | - | 9.8 | pEC50 | - | - | - |
Mol Pharmacol (2007) 72: 1359-68 [PMID:17717109]; Naunyn Schmiedebergs Arch Pharmacol (2006) 373: 158-68 [PMID:16601951] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
