RN1747 [Ligand Id: 4295] activity data from GtoPdb

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  • TRPV4 in Human [GtoPdb: 510] [UniProtKB: Q9HBA0]
  • TRPV4 in Mouse [GtoPdb: 510] [UniProtKB: Q9EPK8]
  • TRPV4 in Rat [GtoPdb: 510] [UniProtKB: Q9ERZ8]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPV4 in Human [GtoPdb: 510] [UniProtKB: Q9HBA0]
GtoPdb - - 6.1 pEC50 770 nM EC50 Biochem Biophys Res Commun (2009) 389: 490-4 [PMID:19737537]
TRPV4 in Mouse [GtoPdb: 510] [UniProtKB: Q9EPK8]
GtoPdb - - 5.4 pEC50 - - - Biochem Biophys Res Commun (2009) 389: 490-4 [PMID:19737537]
TRPV4 in Rat [GtoPdb: 510] [UniProtKB: Q9ERZ8]
GtoPdb - - 5.4 pEC50 - - - Biochem Biophys Res Commun (2009) 389: 490-4 [PMID:19737537]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.