ChEMBL ligand: CHEMBL422420 (ONO-4057)
BLT1 receptor/Leukotriene B4 receptor 1 in Human [ChEMBL: CHEMBL3911] [GtoPdb: 267] [UniProtKB: Q15722] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
BLT1 receptor/Leukotriene B4 receptor 1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3911] [GtoPdb: 267] [UniProtKB: Q15722]
ChEMBL	Binding affinity at leukotriene B4 receptor on intact human PMNs by displacement of [3H]LTB4.	B	8.4	pKi	4	nM	Ki	J Med Chem (1994) 37: 3327-3336 [PMID:7932560]
ChEMBL	Binding affinity against LTB4 receptors in human PMNs using [3H]LTB4 as radioligand	B	8.4	pKi	4	nM	Ki	J Med Chem (1993) 36: 2703-2705 [PMID:8410983]
GtoPdb	-	-	8.43	pKi	3.7	nM	Ki	Prostaglandins (1992) 44: 261-75 [PMID:1332129]
ChEMBL	Compound was tested for inhibitory activity against human neutrophil LTB4 receptor binding	B	8.43	pKi	3.7	nM	Ki	J Med Chem (1996) 39: 2629-2654 [PMID:8709092]
GtoPdb	-	-	6.15	pIC50	700	nM	IC50	Prostaglandins (1992) 44: 261-75 [PMID:1332129]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]