oleoyl-thiophosphate [Ligand Id: 6983] activity data from GtoPdb

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  • LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633]
  • LPA1 receptor in Mouse [GtoPdb: 272] [UniProtKB: P61793]
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  • LPA2 receptor in Mouse [GtoPdb: 273] [UniProtKB: Q9JL06]
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  • LPA3 receptor in Mouse [GtoPdb: 274] [UniProtKB: Q9EQ31]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633]
GtoPdb - - 6.71 pEC50 193 nM EC50 J Med Chem (2005) 48: 4919-30 [PMID:16033271]
LPA1 receptor in Mouse [GtoPdb: 272] [UniProtKB: P61793]
GtoPdb - - 6.71 pEC50 193 nM EC50 Acta Pharmacol Sin (2010) 31: 1213-22 [PMID:20729877]
LPA2 receptor in Mouse [GtoPdb: 273] [UniProtKB: Q9JL06]
GtoPdb - - 6.61 pEC50 244 nM EC50 J Med Chem (2005) 48: 4919-30 [PMID:16033271]
LPA3 receptor in Mouse [GtoPdb: 274] [UniProtKB: Q9EQ31]
GtoPdb - - 6.26 pEC50 546 nM EC50 J Med Chem (2005) 48: 4919-30 [PMID:16033271]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.