MS417 [Ligand Id: 7512] activity data from GtoPdb

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  • bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
GtoPdb Inhibition of MS417 binding to recombinant BRD4-BD1 using FITC-labeled MS417 as the assay probe. - 7.52 pIC50 30 nM IC50 J Biol Chem (2012) 287: 28840-51 [PMID:22645123]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.