CCG-4986 [Ligand Id: 8721] activity data from GtoPdb

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  • regulator of G-protein signaling 4 in Human [GtoPdb: 2811] [UniProtKB: P49798]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
regulator of G-protein signaling 4 in Human [GtoPdb: 2811] [UniProtKB: P49798]
GtoPdb Inhibition of Gαo binding. - 5.38 pIC50 4200 nM IC50 Mol Pharmacol (2007) 71: 169-75 [PMID:17012620];
Mol Pharmacol (2010) 78: 360-5 [PMID:20530129];
Biochim Biophys Acta (2007) 1774: 1213-20 [PMID:17660054]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.