MS023 [Ligand Id: 8955] activity data from GtoPdb

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  • protein arginine methyltransferase 1 in Human [GtoPdb: 1252] [UniProtKB: Q99873]
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  • protein arginine methyltransferase 3 in Human [GtoPdb: 1254] [UniProtKB: O60678]
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  • coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55]
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  • protein arginine methyltransferase 6 in Human [GtoPdb: 1257] [UniProtKB: Q96LA8]
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  • protein arginine methyltransferase 8 in Human [GtoPdb: 1259] [UniProtKB: Q9NR22]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
protein arginine methyltransferase 1 in Human [GtoPdb: 1252] [UniProtKB: Q99873]
GtoPdb - - 7.96 pKi 11 nM Ki ACS Chemical Biology (2015) :
protein arginine methyltransferase 3 in Human [GtoPdb: 1254] [UniProtKB: O60678]
GtoPdb - - 7.26 pKi 55 nM Ki ACS Chemical Biology (2015) :
coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55]
GtoPdb - - 7.64 pKi 23 nM Ki ACS Chemical Biology (2015) :
protein arginine methyltransferase 6 in Human [GtoPdb: 1257] [UniProtKB: Q96LA8]
GtoPdb - - 8.22 pKd 6 nM Kd ACS Chemical Biology (2015) :
GtoPdb - - 9.1 pKi 0.8 nM Ki ACS Chemical Biology (2015) :
protein arginine methyltransferase 8 in Human [GtoPdb: 1259] [UniProtKB: Q9NR22]
GtoPdb - - 8.89 pKi 1.3 nM Ki ACS Chemical Biology (2015) :

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.