probe 1.1 [PMID: 24187130] [Ligand Id: 9191] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145] | ||||||||
| GtoPdb | - | - | 9.6 | pKi | 0.25 | nM | Ki | J Biol Chem (2013) 288: 36703-16 [PMID:24187130] |
| GtoPdb | Measuring βarrestin2 recruitment | - | 5.38 | pEC50 | 4129 | nM | EC50 | J Biol Chem (2013) 288: 36703-16 [PMID:24187130] |
| GtoPdb | Measuring [35S]GTPγS binding | - | 7.51 | pEC50 | 31 | nM | EC50 | J Biol Chem (2013) 288: 36703-16 [PMID:24187130] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
