TAK-828F [Ligand Id: 9867] activity data from GtoPdb

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  • RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449]
GtoPdb Binding to human RORγt isoform. - 8.72 pIC50 1.9 nM IC50 J Med Chem (2018) 61: 2973-2988 [PMID:29510038]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.