bromodomain PHD finger transcription factor

Target id: 2723

Nomenclature: bromodomain PHD finger transcription factor

Family: Non-enzymatic BRD containing proteins

Annotation status:  image of a grey circle Awaiting annotation/under development. Please contact us if you can help with annotation.  » Email us

   GtoImmuPdb view: OFF :     Currently no data for bromodomain PHD finger transcription factor in GtoImmuPdb

Gene and Protein Information
Species TM AA Chromosomal Location Gene Symbol Gene Name Reference
Human - 2903 17q24 BPTF bromodomain PHD finger transcription factor
Mouse - 2921 11 E1 Bptf bromodomain PHD finger transcription factor
Rat - - 10q32.1 Bptf bromodomain PHD finger transcription factor
Previous and Unofficial Names
FAC1 | FALZ
Database Links
CATH/Gene3D
Ensembl Gene
Entrez Gene
GenitoUrinary Development Molecular Anatomy Project
Human Protein Atlas
KEGG Gene
OMIM
RefSeq Nucleotide
RefSeq Protein
UniProtKB
Wikipedia

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Inhibitors
Key to terms and symbols View all chemical structures Click column headers to sort
Ligand Sp. Action Affinity Units Reference
MS363 Hs Inhibition 5.8 pKi 1
pKi 5.8 (Ki 1.62x10-6 M) [1]

References

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1. Zhang G, Plotnikov AN, Rusinova E, Shen T, Morohashi K, Joshua J, Zeng L, Mujtaba S, Ohlmeyer M, Zhou MM. (2013) Structure-guided design of potent diazobenzene inhibitors for the BET bromodomains. J. Med. Chem.56 (22): 9251-64. [PMID:24144283]

How to cite this page

Non-enzymatic BRD containing proteins: bromodomain PHD finger transcription factor. Last modified on 13/02/2017. Accessed on 19/10/2017. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2723.