isotonitazene [Ligand Id: 12955] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372] | ||||||||
| GtoPdb | Potency determined in a cAMP accumulation assay in HEK cells expressing hMOR | - | 10.3 | pEC50 | 0.05 | nM | EC50 | Drug Alcohol Depend (2023) 249: 109939 [PMID:37276825] |
| μ receptor in Rat [GtoPdb: 319] [UniProtKB: P33535] | ||||||||
| GtoPdb | Binding affinity in rat brain | - | 7.95 | pKi | 11.2 | nM | Ki | Drug Alcohol Depend (2023) 249: 109939 [PMID:37276825] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
